{"id":2269,"date":"2023-03-31T08:12:51","date_gmt":"2023-03-31T11:12:51","guid":{"rendered":"https:\/\/ibyme.org.ar\/investigacion\/?page_id=2269"},"modified":"2023-06-20T20:55:26","modified_gmt":"2023-06-20T23:55:26","slug":"lineas-de-investigacion-oncologia","status":"publish","type":"page","link":"https:\/\/ibyme.org.ar\/investigacion\/laboratorios\/patologia-y-farmacologia-molecular\/lineas-de-investigacion-oncologia\/","title":{"rendered":"L\u00edneas de Investigaci\u00f3n: Oncolog\u00eda"},"content":{"rendered":"<p><div class=\"fusion-fullwidth fullwidth-box fusion-builder-row-1 fusion-flex-container has-pattern-background has-mask-background fusion-parallax-none hundred-percent-fullwidth non-hundred-percent-height-scrolling\" 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class=\"fusion-title-heading title-heading-left\" style=\"margin:0;\">Patolog\u00eda y Farmacolog\u00eda Molecular<\/h1><\/div><\/div><\/div><\/div><\/div><div class=\"fusion-fullwidth fullwidth-box fusion-builder-row-4 fusion-flex-container has-pattern-background has-mask-background nonhundred-percent-fullwidth non-hundred-percent-height-scrolling\" style=\"--awb-border-radius-top-left:0px;--awb-border-radius-top-right:0px;--awb-border-radius-bottom-right:0px;--awb-border-radius-bottom-left:0px;--awb-flex-wrap:wrap;\" ><div class=\"fusion-builder-row fusion-row fusion-flex-align-items-flex-start fusion-flex-content-wrap\" style=\"max-width:1248px;margin-left: calc(-4% \/ 2 );margin-right: calc(-4% \/ 2 );\"><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-2 fusion_builder_column_1_1 1_1 fusion-flex-column\" style=\"--awb-bg-size:cover;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:1.92%;--awb-margin-bottom-large:20px;--awb-spacing-left-large:1.92%;--awb-width-medium:100%;--awb-order-medium:0;--awb-spacing-right-medium:1.92%;--awb-spacing-left-medium:1.92%;--awb-width-small:100%;--awb-order-small:0;--awb-spacing-right-small:1.92%;--awb-spacing-left-small:1.92%;\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-title title fusion-title-2 fusion-sep-none fusion-title-text fusion-title-size-two\" style=\"--awb-text-color:var(--awb-color5);--awb-font-size:22px;\"><h2 class=\"fusion-title-heading title-heading-left\" style=\"font-family:&quot;Red Hat Display&quot;;font-style:normal;font-weight:700;margin:0;font-size:1em;\">L\u00edneas de Investigaci\u00f3n: Oncolog\u00eda<\/h2><\/div><\/div><\/div><\/div><\/div><div class=\"fusion-fullwidth fullwidth-box fusion-builder-row-5 fusion-flex-container has-pattern-background has-mask-background nonhundred-percent-fullwidth non-hundred-percent-height-scrolling\" style=\"--awb-border-radius-top-left:0px;--awb-border-radius-top-right:0px;--awb-border-radius-bottom-right:0px;--awb-border-radius-bottom-left:0px;--awb-flex-wrap:wrap;\" ><div class=\"fusion-builder-row fusion-row fusion-flex-align-items-flex-start fusion-flex-content-wrap\" style=\"max-width:1248px;margin-left: calc(-4% \/ 2 );margin-right: calc(-4% \/ 2 );\"><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-3 fusion_builder_column_1_1 1_1 fusion-flex-column\" style=\"--awb-bg-size:cover;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:1.92%;--awb-margin-bottom-large:20px;--awb-spacing-left-large:1.92%;--awb-width-medium:100%;--awb-order-medium:0;--awb-spacing-right-medium:1.92%;--awb-spacing-left-medium:1.92%;--awb-width-small:100%;--awb-order-small:0;--awb-spacing-right-small:1.92%;--awb-spacing-left-small:1.92%;\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-text fusion-text-1\"><p>Receptores a histamina: transducci\u00f3n de se\u00f1ales y mecanismos de acci\u00f3n de ligandos.<br \/>\nLa histamina ejerce m\u00faltiples acciones mediante la interacci\u00f3n con cuatro receptores espec\u00edficos, (H1-H4) pertenecientes a la superfamilia de receptores acoplados a prote\u00ednas G (GPCRs). Antagonistas\/agonistas inversos de los receptores H1 y H2 son ampliamente utilizados para el tratamiento de alergias y acidez g\u00e1strica, respectivamente, y de hecho se encuentran entre las veinte drogas de venta libre y bajo receta m\u00e1s consumidas a nivel mundial. Durante los \u00faltimos a\u00f1os, nuestro laboratorio ha realizado numerosos aportes sobre la se\u00f1alizaci\u00f3n y regulaci\u00f3n de la respuesta celular a trav\u00e9s de los receptores H1 y H2 a histamina. Recientemente hemos demostrado la existencia de una regulaci\u00f3n cruzada a nivel de dichos receptores inducida tanto por sus agonistas como por sus antagonistas\/agonistas inversos. Nuestro pr\u00f3ximo paso ser\u00e1 analizar los mecanismos involucrados en esta regulaci\u00f3n, as\u00ed como su relevancia terap\u00e9utica en diferentes modelos de estudio. De esta manera, aportaremos nuevas bases para la utilizaci\u00f3n racional de agonistas o antagonistas histamin\u00e9rgicos en distintas patolog\u00edas, para el desarrollo de nuevos f\u00e1rmacos y para el planteo de nuevas estrategias terap\u00e9uticas en estudios de reposicionamiento de drogas.<\/p>\n<p>Blancos terap\u00e9uticos asociados a la cascada del AMPc en leucemias mieloides humanas.<br \/>\nUn enfoque potencialmente menos t\u00f3xico para el tratamiento de la leucemia mieloide aguda es la denominada \u00abterapia diferenciante\u00bb. Esta terapia se basa en el hecho de que las c\u00e9lulas neopl\u00e1sicas exhiben frecuentemente defectos reversibles en el proceso de diferenciaci\u00f3n. Por lo tanto, con un tratamiento apropiado puede eventualmente lograrse la reprogramaci\u00f3n de dichas c\u00e9lulas, disminuyendo su capacidad proliferativa e induciendo su maduraci\u00f3n o su muerte por apoptosis. Hemos demostrado previamente que el balance entre la producci\u00f3n, degradaci\u00f3n y exclusi\u00f3n de AMPc es esencial para la proliferaci\u00f3n\/diferenciaci\u00f3n de c\u00e9lulas leuc\u00e9micas. Diferentes mol\u00e9culas participan en esta regulaci\u00f3n, incluyendo al receptor H2 a histamina, a la quinasa responsable de la desensibilizaci\u00f3n del receptor H2 a histamina GRK2, a las fosfodiesterasas y al transportador de AMPc MRP4, entre otras. En este sentido, nos interesa evaluar el efecto conjunto de la activaci\u00f3n del rH2 e inhibici\u00f3n farmacol\u00f3gica de MRP4 y\/o GRK2 sobre la proliferaci\u00f3n\/diferenciaci\u00f3n celular, en modelos in vitro e in vivo de leucemias mieloides humanas. Si bien estos blancos moleculares asociados a la cascada del AMPc han sido estudiados en profundidad por nuestro laboratorio y demostrada su asociaci\u00f3n con el deseado proceso de inducci\u00f3n de diferenciaci\u00f3n celular, al presente no existen estudios que permitan postular su acci\u00f3n sin\u00e9rgica o la posible aplicaci\u00f3n de estrategias polifarmacol\u00f3gicas en la terapia diferenciante.<\/p>\n<p>Asimismo, colaboramos estrechamente con laboratorios del ININFA-UBA-CONICET del \u00c1rea de Oncolog\u00eda Molecular en l\u00edneas relacionadas a tumores de p\u00e1ncreas y ves\u00edcula biliar.<\/p>\n<\/div><\/div><\/div><\/div><\/div><\/p>\n","protected":false},"excerpt":{"rendered":"","protected":false},"author":12,"featured_media":0,"parent":2266,"menu_order":2,"comment_status":"closed","ping_status":"closed","template":"100-width.php","meta":{"_acf_changed":false,"inline_featured_image":false,"wpupg_custom_link":[],"wpupg_custom_link_behaviour":["default"],"wpupg_custom_link_nofollow":[],"wpupg_custom_image":[],"wpupg_custom_image_id":[],"footnotes":""},"page_category":[],"class_list":["post-2269","page","type-page","status-publish","hentry"],"acf":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v26.6 - 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